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DCC-2036

DCC-2036 (Rebastinib) is a highly potent, non-ATP-competitive BCR-ABL1 inhibitor with IC50 of 0.8 and 4 nM for native ABL1 and gatekeeper mutant ABL1 T315I, respectively.

Product Specifications

CAS Number

1020172-07-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

553.5869

Molecular Formula

C30H28FN7O3

Notes

Research use only, not for human use.

Receptor

Abl1|FLT3|p-Abl1 (native) |p-Abl1 (T315I) |u-Abl1 (native)

Available Sizes

Curated Selection

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