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CLK inhibitor 2

A potent, selective inhibitor of cdc2-like kinase CLK1 and CLK2 with IC50 of 1.1 and 2.4 nM, respectively; moderately inhibits PI3Kα, and >100-fold selectivity over SRPK1/2/3.

Product Specifications

CAS Number

1005776-20-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

360.421

Molecular Formula

C20H20N6O

Notes

Research use only, not for human use.

Receptor

CLK

Available Sizes

Frequently Asked Questions

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