CY 208-243

CY 208-243 is a selective dopamine D1 receptor agonist which exhibits antiparkinsonian activity[1].

Product Specifications

CAS Number

[100999-26-6]

UNSPSC

12352005

Target

Dopamine Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neurodegeneration

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/cy-208-243.html

Purity

99.99

Solubility

DMSO : 50 mg/mL (ultrasonic)

Smiles

CN1[C@@](C2)([H])[C@@](C3=CC=CC=C3C1)([H])C4=CC=CC5=C4C2=CN5

Molecular Formula

C19H18N2

Molecular Weight

274.36

References & Citations

[1]Imperato A, et al. CY 208-243, a novel dopamine D-1 receptor agonist, fails to modify dopamine release in freely moving rats. Eur J Pharmacol. 1989 Jan 24;160 (1) :155-8.|[2]Temlett JA, et al. The D-1 dopamine receptor partial agonist, CY 208-243, exhibits antiparkinsonian activity in the MPTP-treated marmoset. Eur J Pharmacol. 1988 Nov 1;156 (2) :197-206.