FL104

FL104 is a potent small molecule urotensin II receptor agonist with pEC50 of 7.11 for UTII receptor in R-SATTM assay[1][2].

Product Specifications

CAS Number

[885672-81-1]

UNSPSC

12352005

Target

Others

Type

Reference compound

Related Pathways

Others

Field of Research

Others

Assay Protocol

https://www.medchemexpress.com/fl104.html

Solubility

10 mM in DMSO

Smiles

O=C(C1=CC=C(C2=CC=CC=C2)C=C1)NC(CCN(C)C)C3=CC=C(C=C3)Cl

Molecular Formula

C24H25ClN2O

Molecular Weight

392.92

References & Citations

[1]Lehmann F, et al. Novel and potent small-molecule urotensin II receptor agonists. Bioorg Med Chem. 2009 Jul 1;17 (13) :4657-65.|[2]Lehmann F, et al. Design, parallel synthesis and SAR of novel urotensin II receptor agonists. Eur J Med Chem. 2007 Feb;42 (2) :276-85.