PD-149164
PD-149164 is a potent agonist of cholecystokinin B (CCK-B) receptor, with IC50 values of 0.083 nM and 75 nM in binding assay to CCK-B and CCK-A[1].
Product Specifications
CAS Number
181941-32-2
UNSPSC
12352005
Target
Cholecystokinin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Endocrinology; Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/pd-149164.html
Smiles
O=C(C[C@H](CC1=CC=C(C=C1)F)NC([C@@](NC(OC2C3CC4CC(CC2C4)C3)=O)(C)CC5=CNC6=C5C=CC=C6)=O)O
Molecular Formula
C33H38FN3O5
Molecular Weight
575.67
References & Citations
[1]J Hughes, et al. Characterization of novel peptoid agonists for the CCK-A receptor. Regul Pept. 1996 Aug 27;65 (1) :15-21.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CCKAR; CCKBR
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS6172893-01 0.1 mL
CORO1B (coronin, Actin Binding Protein, 1B, CORONIN-2, DKFZp762I166) (Biotin)
Sign In for Pricing
View Details MBS6172893-02 5x 0.1 mL
CORO1B (coronin, Actin Binding Protein, 1B, CORONIN-2, DKFZp762I166) (Biotin)
Sign In for Pricing
View Details 
NBP2-98155AF532 0.1 mL
Rabbit Polyclonal SLC16A4 Antibody [Alexa Fluor 532]
Sign In for Pricing
View Details K7328006 1.0 µg DNA
LOC361016 sgRNA CRISPR/Cas9 All-in-One Lentivector (Rat) (Target 1)
Sign In for Pricing
View Details