PD-149164
PD-149164 is a potent agonist of cholecystokinin B (CCK-B) receptor, with IC50 values of 0.083 nM and 75 nM in binding assay to CCK-B and CCK-A[1].
Product Specifications
CAS Number
[181941-32-2]
UNSPSC
12352005
Target
Cholecystokinin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Endocrinology; Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/pd-149164.html
Smiles
O=C(C[C@H](CC1=CC=C(C=C1)F)NC([C@@](NC(OC2C3CC4CC(CC2C4)C3)=O)(C)CC5=CNC6=C5C=CC=C6)=O)O
Molecular Formula
C33H38FN3O5
Molecular Weight
575.67
References & Citations
[1]J Hughes, et al. Characterization of novel peptoid agonists for the CCK-A receptor. Regul Pept. 1996 Aug 27;65 (1) :15-21.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CCKAR; CCKBR
Curated Selection
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