Cebranopadol ((1α,4α)stereoisomer)
Product Specifications
CAS Number
863513-93-3
UNSPSC Description
Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol. Cebranopadol is a potent agonist activity on ORL-1.
Target Antigen
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein;Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/Cebranopadol-_1_alpha_,4_alpha__stereoisomer.html
Solubility
DMSO : < 1 mg/mL (ultrasonic;warming;heat to 60°C)|H2O : < 0.1 mg/mL (ultrasonic;warming;heat to 60°C)
Smiles
CN(C)[C@@]1(C2=CC=CC=C2)CC[C@]3(C(N4)=C(CCO3)C5=C4C=CC(F)=C5)CC1
Molecular Weight
378.48
References & Citations
[1]Schunk S, et al. Discovery of a Potent Analgesic NOP and Opioid Receptor Agonist: Cebranopadol. ACS Med Chem Lett. 2014 Jun 24;5(8):857-62
Shipping Conditions
Room Temperature
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
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