LUF5981
LUF5981 is a relatively potent adenosine A2A receptor (A2A) antagonist with pIC50 value of 6.7[1].
Product Specifications
CAS Number
[929641-63-4]
UNSPSC
12352005
Target
Adenosine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/luf5981.html
Smiles
C12=NC(C3=CC=CC=C3)=CC(C4=CC=CC=C4)=C1N=C(C5CCCCC5)N2
Molecular Formula
C24H23N3
Molecular Weight
353.46
References & Citations
[1]Fan Fan, et al. The integration of pharmacophore-based 3D QSAR modeling and virtual screening in safety profiling: A case study to identify antagonistic activities against adenosine receptor, A2A, using 1,897 known drugs. PLoS One. 2019 Jan 3;14 (1) :e0204378.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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