Glucagon receptor antagonist-3
Glucagon receptor antagonist-3 is a highly potent glucagon receptor antagonist.
Product Specifications
CAS Number
[202917-17-7]
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H335
Target
GCGR
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-sugar/lipid metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/glucagon-receptor-antagonists-3.html
Concentration
10mM
Purity
99.78
Solubility
DMSO : ≥ 100 mg/mL
Smiles
CC(C1=NC(C(C)C)=C([C@]([C@]2=CC=C(C=C2O)F)=C1[C@@H](C)O)CCC)C
Molecular Formula
C22H30FNO2
Molecular Weight
359.48
Precautions
H302, H315, H319, H335
References & Citations
[1]Ladouceur, Gaetan H. et al. Integration of optimized substituent patterns to produce highly potent 4-aryl-pyridine glucagon receptor antagonists. Bioorganic & Medicinal Chemistry Letters (2002), 12 (23), 3421-3424.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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