VU0240382
VU0240382 is a metabotropic glutamate receptor subtype 5 modulator whose activity differs depending on whether it has allosteric agonist activity. VU0240382 with allosteric agonist activity can activate mGlu (5) receptors in cell lines, but has no agonist activity in natural systems and has similar efficacy to mGlu (5) modulators without allosteric agonist activity in animal models.
Product Specifications
CAS Number
[1092550-36-1]
UNSPSC
12352005
Target
Others
Type
Reference compound
Related Pathways
Others
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/vu0240382.html
Smiles
O=C1NCCC2=C1C=CC(C#CC3=CC=CC=C3)=C2
Molecular Formula
C17H13NO
Molecular Weight
247.29
References & Citations
[1]Functional impact of allosteric agonist activity of selective positive allosteric modulators of metabotropic glutamate receptor subtype 5 in regulating central nervous system function
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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