Capeserod (hydrochloride)
Capeserod hydrochloride (SL65.0155) is a 5-HT4 (e) receptor partial agonist (Ki=0.6 nM) with potent cognitive enhancing properties. Capeserod hydrochloride acts as a partial agonist in cells expressing 5-HT4 (b) and 5-HT4 (e) splice variants, stimulating cAMP production with IC50 values of 244 and 29 nM, respectively. Capeserod hydrochloride is used in the study of memory impairment and dementia[1].
Product Specifications
CAS Number
191023-43-5
Product Name Alternative
SL65.0155
UNSPSC
12352005
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/capeserod-hydrochloride.html
Smiles
O=C1OC(C2=C3OCCOC3=C(N)C(Cl)=C2)=NN1C4CCN(CC4)CCC5=CC=CC=C5.Cl
Molecular Formula
C23H26Cl2N4O4
Molecular Weight
493.38
References & Citations
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
5-HT4 Receptor; Apolipoprotein D
Frequently Asked Questions
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