CP-293019
CP-293019 is a dopamine D4 receptor antagonist, with a Ki value of 3.4 nM. CP-293019 can inhibit Apomorphine induced hyperactivity in rats[1].
Product Specifications
CAS Number
179089-90-8
UNSPSC
12352005
Target
Dopamine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cp-293019.html
Smiles
FC1=CN=C(N2C[C@](CC[C@@H](COC3=CC=C(F)C=C3)C4)([H])N4CC2)N=C1
Molecular Formula
C19H22F2N4O
Molecular Weight
360.40
References & Citations
[1]Sanner MA, et al. Synthesis, SAR and pharmacology of CP-293,019: a potent, selective dopamine D4 receptor antagonist. Bioorg Med Chem Lett. 1998 Apr 7;8 (7) :725-30.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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