Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

PDE4-IN-18

PDE4-IN-18 (compound 1l) is a PDE4 inhibitor (IC50=1.55 μM) with anti-inflammatory activity. PDE4-IN-18 exerts anti-inflammatory effects by reducing excessive immune cell infiltration and intestinal membrane formation, as well as reducing the mRNA expression of pro-inflammatory cytokines (such as TNF-α and IL-6) in synovial tissue. PDE4-IN-18 can be used in the study of rheumatoid arthritis and psoriasis[1].

Product Specifications

UNSPSC

12352211

Target

Interleukin Related; Phosphodiesterase (PDE) ; TNF Receptor

Type

Reference compound

Related Pathways

Apoptosis; Immunology/Inflammation; Metabolic Enzyme/Protease

Field of Research

Inflammation/Immunology

Assay Protocol

https://www.medchemexpress.com/pde4-in-18.html

Smiles

O=C1C2=CC(F)=CC=C2C(CC=C)=C(C3=CC(NS(=O)(C4=CC=CC=C4)=O)=CC=C3)N1

Molecular Formula

C24H19FN2O3S

Molecular Weight

434.48

References & Citations

[1]Bhuktar, et al. "Targeting next-generation PDE4 inhibitors in search of potential management of rheumatoid arthritis and psoriasis." Bioorganic Chemistry (2024) : 107689.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

PDE4

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Liver Carboxylesterase 1 Antibody
KC-3311-01 50 μL

Liver Carboxylesterase 1 Antibody

Sign In for Pricing
View Details
Liver Carboxylesterase 1 Antibody
KC-3311-02 100 µL

Liver Carboxylesterase 1 Antibody

Sign In for Pricing
View Details
Liver Carboxylesterase 1 Antibody
KC-3311-03 1 mL

Liver Carboxylesterase 1 Antibody

Sign In for Pricing
View Details
Elab Fluor® 700 Anti-Mouse CD16/32 Antibody[2.4G2]
E-AB-F0997UM1-01 25 µg

Elab Fluor® 700 Anti-Mouse CD16/32 Antibody[2.4G2]

Sign In for Pricing
View Details
Elab Fluor® 700 Anti-Mouse CD16/32 Antibody[2.4G2]
E-AB-F0997UM1-02 100 µg

Elab Fluor® 700 Anti-Mouse CD16/32 Antibody[2.4G2]

Sign In for Pricing
View Details
ω-Hydroxy-DEET-D10 (>80%)
TRC-H934204-1MG 1 mg

ω-Hydroxy-DEET-D10 (>80%)

Sign In for Pricing
View Details