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CPI-203

CPI-203 is a primary amide analog of (+) -JQ1, which has shown superior bioavailability with oral or i.p. administration. CPI-203 downregulates Myc expression, causes G1 cell cycle arrest and attenuates cell proliferation in human pancreatic neuroendocrine tumors. CPI-203 also arrests the growth of T cell acute lymphoblastic leukemia cells in vitro (EC50= 91.2 nM) .

Product Specifications

Format

Solid

Molecular Formula

C19H18ClN5OS

Shipping Conditions

Room Temperature

Storage Conditions

At least 6 months at -20°C.

Calculated Molecular Weight

399.9 Da

CAS Number

1446144-04-2

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