Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

Galantide (TFA)

Galantide TFA is a reversible and non-specific galanin (GAL) receptor antagonist. Galantide TFA dose-dependently shows antagonism to galanin-induced K+ conductance with an IC50 value of 4 nM. Galantide TFA can be used for the research of neurological disease and hormone metabolism research[1][2].

Product Specifications

CAS Number

9007-83-4

UNSPSC

12352209

Target

Neuropeptide Y Receptor

Type

Peptides

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Metabolic Disease; Neurological Disease

Assay Protocol

https://www.medchemexpress.com/galantide-tfa.html

Purity

98.09

Solubility

DMSO : 100 mg/mL (ultrasonic) |H2O : < 0.1 mg/mL (ultrasonic; adjust pH to 2 with HCl)

Smiles

OC(C(F)(F)F)=O.OC(C=C1)=CC=C1C[C@@H](C(N[C@@H](CC(C)C)C(N[C@@H](CC(C)C)C(NCC(N2[C@@H](CCC2)C(N[C@@H](CCC(N)=O)C(N[C@@H](CCC(N)=O)C(N[C@H](C(N[C@H](C(NCC(N[C@@H](CC(C)C)C(N[C@H](C(N)=O)CCSC)=O)=O)=O)CC3=CC=CC=C3)=O)CC4=CC=CC=C4)=O)=O)=O)=O)=O)=O)=O)NC(CNC([C@H](C)NC([C@H](CO)NC([C@H](CC(N)=O)NC([C@H](CC(C)C)NC([C@H]([C@H](O)C)NC([C@@H](NC(CN)=O)CC5=CNC6=CC=CC=C56)=O)=O)=O)=O)=O)=O)=O

Molecular Formula

C106H152F3N25O28S

Molecular Weight

2313.55

References & Citations

[1]Mulvaney JM, et al. Galantide distinguishes putative subtypes of galanin receptors in mudpuppy parasympathetic neurons. Eur J Pharmacol. 1995 Dec 4;287 (1) :97-100.|[2]Sahu A, et al. Role of galanin in stimulation of pituitary luteinizing hormone secretion as revealed by a specific receptor antagonist, galantide. Endocrinology. 1994 Feb;134 (2) :529-36.

Shipping Conditions

Blue Ice

Storage Conditions

-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture and light, under nitrogen)

Scientific Category

Peptides

Clinical Information

No Development Reported

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Anti-West Nile Virus (WNV) (lineage 1, strain NY99) NS1 Polyclonal Antibody
E-AB-V1326-01 20 µL

Anti-West Nile Virus (WNV) (lineage 1, strain NY99) NS1 Polyclonal Antibody

Sign In for Pricing
View Details
Anti-West Nile Virus (WNV) (lineage 1, strain NY99) NS1 Polyclonal Antibody
E-AB-V1326-02 100 µL

Anti-West Nile Virus (WNV) (lineage 1, strain NY99) NS1 Polyclonal Antibody

Sign In for Pricing
View Details
Etaphos
TRC-E825960-500MG 500 mg

Etaphos

Sign In for Pricing
View Details
RAB23 (NM_016277) Human Over-expression Lysate
LC402532 20 µg

RAB23 (NM_016277) Human Over-expression Lysate

Sign In for Pricing
View Details
Pivaloylglycine-13C2,15N
TRC-P550738-5MG 5 mg

Pivaloylglycine-13C2,15N

Sign In for Pricing
View Details
ATP2A1 Human Gene Knockout Kit (CRISPR)
KN414911 1 Kit

ATP2A1 Human Gene Knockout Kit (CRISPR)

Sign In for Pricing
View Details