GV150013X
GV150013X is an antagonist for cholecystokinin-2/gastrin receptor (CCK2R), with Ki of 2.29 nM. GV150013X attenuates central nervous disorders, such as anxiety and panic disorder[1].
Product Specifications
CAS Number
151386-96-8
UNSPSC
12352005
Target
Cholecystokinin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/gv150013x.html
Solubility
10 mM in DMSO
Smiles
O=C([C@H](C1=O)NC(NC2=CC=CC=C2)=O)N(C3=CC=CC=C3)C4=CC=CC=C4N1CC5(C[C@@H]6C7)C[C@@H]7C[C@@H](C6)C5
Molecular Formula
C33H34N4O3
Molecular Weight
534.65
References & Citations
[1]Novak D, et al., CCK2R antagonists: from SAR to clinical trials. Drug Discov Today. 2020 Aug;25 (8) :1322-1336.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CCKBR
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
LC401148 20 µg
Ceramide glucosyltransferase (UGCG) (NM_003358) Human Over-expression Lysate
Sign In for Pricing
View Details 
PKSQ050018-01 10 µg
Recombinant Cynomolgus B7-1/CD80 Protein (Fc Tag)
Sign In for Pricing
View Details PKSQ050018-02 50 µg
Recombinant Cynomolgus B7-1/CD80 Protein (Fc Tag)
Sign In for Pricing
View Details 
