GV150013X
GV150013X is an antagonist for cholecystokinin-2/gastrin receptor (CCK2R), with Ki of 2.29 nM. GV150013X attenuates central nervous disorders, such as anxiety and panic disorder[1].
Product Specifications
CAS Number
151386-96-8
UNSPSC
12352005
Target
Cholecystokinin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/gv150013x.html
Solubility
10 mM in DMSO
Smiles
O=C([C@H](C1=O)NC(NC2=CC=CC=C2)=O)N(C3=CC=CC=C3)C4=CC=CC=C4N1CC5(C[C@@H]6C7)C[C@@H]7C[C@@H](C6)C5
Molecular Formula
C33H34N4O3
Molecular Weight
534.65
References & Citations
[1]Novak D, et al., CCK2R antagonists: from SAR to clinical trials. Drug Discov Today. 2020 Aug;25 (8) :1322-1336.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CCKBR
Available Sizes
Frequently Asked Questions
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