OPC-51803

OPC-51803 is an orally active nonpeptide vasopressin V2 receptor agonist. OPC-51803 can be used for the research of micturition disorders that result in frequent micturition, such as that from polyuria, nocturnal polyuria, and some kinds of urinary incontinence[1].

Product Specifications

CAS Number

[192514-54-8]

UNSPSC

12352005

Target

Vasopressin Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Metabolic Disease

Assay Protocol

https://www.medchemexpress.com/opc-51803.html

Purity

99.77

Solubility

DMSO : 100 mg/mL (ultrasonic)

Smiles

O=C(N1CCC[C@H](CC(NC(C)C)=O)C2=CC=CC=C21)C3=CC=C(N4CCCC4)C=C3Cl

Molecular Formula

C26H32ClN3O2

Molecular Weight

454.00

References & Citations

[1]Nakamura S, et al. Effects of OPC-51803, a novel, nonpeptide vasopressin V2-receptor agonist, on micturition frequency in Brattleboro and aged rats. J Pharmacol Sci. 2003 Dec;93 (4) :484-8.