Tiapride (hydrochloride) (Standard)

Tiapride (hydrochloride) (Standard) is the analytical standard of Tiapride (hydrochloride) . This product is intended for research and analytical applications. Tiapride hydrochloride is a selective and orally active D2 and D3 dopamine receptors antagonist with IC50 values of 110-320 nM and 180 nM, respectively. Tiapride hydrochloride shows anti-dyskinetic activity and anxiolytic activity. Tiapride hydrochloride is a neuroleptic agent[1][2].

Product Specifications

CAS Number

[51012-33-0]

UNSPSC

12352005

Target

Dopamine Receptor; Reference Standards

Type

Reference Standards

Related Pathways

GPCR/G Protein; Neuronal Signaling; Others

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/tiapride-hydrochloride-standard.html

Smiles

O=C(NCCN(CC)CC)C1=CC(S(=O)(C)=O)=CC=C1OC.[H]Cl

Molecular Formula

C15H25ClN2O4S

Molecular Weight

364.89

References & Citations

[1]Scatton B, et al. The preclinical pharmacologic profile of tiapride. Eur Psychiatry. 2001 Jan;16 Suppl 1:29s-34s.|[2]Peters DH, et al. Tiapride. A review of its pharmacology and therapeutic potential in the management of alcohol dependence syndrome. Drugs. 1994 Jun;47 (6) :1010-32.