EHMT2-IN-2

EHMT2-IN-2 is a potent EHMT inhibitor, with IC50s of all [1].

Product Specifications

CAS Number

[2230850-47-0]

UNSPSC

12352005

Target

Histone Methyltransferase

Type

Reference compound

Related Pathways

Epigenetics

Applications

Neuroscience-Neuromodulation

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/ehmt2-in-2.html

Concentration

10mM

Purity

99.0

Solubility

DMSO : 50 mg/mL (ultrasonic)

Smiles

CC1=CC(NC)=NC(NC2=CC=C(OC)C(C(N3)=C(C)C4=C3C=NC=C4)=C2)=N1

Molecular Formula

C21H22N6O

Molecular Weight

374.44

References & Citations

[1]John Emmerson Campbell, et al. Amine-substituted heterocyclic compounds as ehmt2 inhibitors and methods of use thereof. WO2018118842A1.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

EHMT1/GLP/KMT1D; EHMT2/G9a/KMT1C

Available Sizes

Curated Selection

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