EHMT2-IN-2
EHMT2-IN-2 is a potent EHMT inhibitor, with IC50s of all [1].
Product Specifications
CAS Number
[2230850-47-0]
UNSPSC
12352005
Target
Histone Methyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Neuroscience-Neuromodulation
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/ehmt2-in-2.html
Concentration
10mM
Purity
99.0
Solubility
DMSO : 50 mg/mL (ultrasonic)
Smiles
CC1=CC(NC)=NC(NC2=CC=C(OC)C(C(N3)=C(C)C4=C3C=NC=C4)=C2)=N1
Molecular Formula
C21H22N6O
Molecular Weight
374.44
References & Citations
[1]John Emmerson Campbell, et al. Amine-substituted heterocyclic compounds as ehmt2 inhibitors and methods of use thereof. WO2018118842A1.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
EHMT1/GLP/KMT1D; EHMT2/G9a/KMT1C
Available Sizes
Curated Selection
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