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TLR9-IN-1

Product Specifications

UNSPSC Description

TLR9-IN-1 is a potent and selective TLR9 inhibitor with an IC50 value of 7 nM for human TLR9. TLR9-IN-1 can be used for researching diseases associated with undesirable immune response[1].

Target Antigen

Toll-like Receptor (TLR)

Type

Reference compound

Related Pathways

Immunology/Inflammation

Applications

COVID-19-immunoregulation

Field of Research

Inflammation/Immunology

Assay Protocol

https://www.medchemexpress.com/tlr9-in-1.html

Solubility

DMSO : 500 mg/mL (ultrasonic)

Smiles

O=C(C1CCN(CC1)C2=NN=CC3=CN(C4=CC=C(C)C=C4)N=C32)NCCCN(C)C

Molecular Weight

421.54

References & Citations

[1]Albert Frederick Candia, et al. Toll-like receptor antagonist compounds and methods of use. WO2018089695

Shipping Conditions

Room Temperature

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-148045/TLR9-IN-1-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-148045/TLR9-IN-1-SDS-MedChemExpress.pdf

Clinical Information

No Development Reported

CAS Number

2226366-86-3

Available Sizes

Curated Selection

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