(E/Z) -VU0029767
(E/Z) -VU0029767 is an allosteric enhancer of M1 muscarinic receptors with the activity to modulate M1 receptor activity. (E/Z) -VU0029767 can enhance M1 receptor activity by increasing agonist affinity, but exhibits different properties from other compounds under different experimental conditions, such as effects on mutant M1 receptors and effects on downstream signaling pathways.
Product Specifications
CAS Number
326001-01-8
UNSPSC
12352005
Hazard Statement
H302-H315-H319-H335-H410
Target
Others
Type
Reference compound
Related Pathways
Others
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/e-z-vu0029767.html
Smiles
O=C(N/N=C/C1=C2C=CC=CC2=CC=C1O)CNC3=CC=C(OCC)C=C3
Molecular Formula
C21H21N3O3
Molecular Weight
363.41
Precautions
P261-P264-P270-P271-P273-P280-P302+P352-P304+P340-P305+P351+P338-P330-P362+P364-P391-P403+P233-P405-P501
References & Citations
[1]Allosteric activators of muscarinic receptors as novel approaches for treatment of CNS disorders
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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