AMPA receptor modulator-2
AMPA receptor modulator-2 (Example 134) is a AMPA receptor modulator, with a pIC50 of 10.1 for TARPγ8 dependent AMPA receptor[1]. pIC50 = -lgIC50.
Product Specifications
CAS Number
[2034181-36-5]
UNSPSC
12352005
Target
IGluR
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/ampa-receptor-modulator-2.html
Purity
98.55
Solubility
DMSO : 250 mg/mL (ultrasonic)
Smiles
O=C1SC2=CC(N3C(C(F)(F)F)=NC4=CC=C(C(F)(F)F)N=C43)=CC=C2N1
Molecular Formula
C15H6F6N4OS
Molecular Weight
404.29
References & Citations
[1]BERRY CYNTHIA G B (US), et al. AZABENZIMIDAZOLES AND THEIR USE AS AMPA RECEPTOR MODULATORS. Patent. WO2016176460.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
AMPA Receptor
Available Sizes
Curated Selection
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