ERAP1-IN-2
ERAP1-IN-2 (compound 3f) is an inhibitor of ERAP1 (endoplasmic reticulum aminopeptidase 1) . ERAP1-IN-2 has an IC50 value of 1.72 μM against hERAP1[1].
Product Specifications
UNSPSC
12352005
Target
Aminopeptidase
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/erap1-in-2.html
Smiles
O=C(O)C1=CC=C(CC(SC(N2)=S)C2=O)C=C1
Molecular Formula
C11H9NO3S2
Molecular Weight
267.32
References & Citations
[1]Fougiaxis V, et al. First fragment-based screening identifies new chemotypes inhibiting ERAP1-metalloprotease. Eur J Med Chem. 2024 Sep 30;280:116926.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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