GAC0001E5
GAC0001E5 (1E5) is a dual LXR inverse agonist and degrader (IC50 = 5.4-9.1 μM in pancreatic cancer cells) . It inhibits tumor growth and induces apoptosis by promoting LXRα/β degradation and suppressing transcriptional activity.
Product Specifications
CAS Number
927969-67-3
Purity
98.89% (May vary between batches)
Smiles
O=C1N=C (NC2=CC=CC (=C2) C (F) (F) F) NC (=C1) C=3C=CC=CC3
Molecular Formula
C17H12F3N3O
Molecular Weight
331.29
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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