What is the catalog number for NEP108?

The catalog number for NEP108 is orb3177182.

What sizes are available for NEP108?

NEP108 is available in the following size(s): 50 mg, 10 mg.

How many pack sizes does NEP108 come in?

NEP108 is available in 2 different pack sizes.

NEP108 is currently made to order / not held in immediate stock. Contact us for lead time.

NEP108

NEP108 is a BRD4 PROTAC degrader designed based on GID4 E3 ligase, with a DC50 of approximately 3.8 μM. It exhibits strong affinity for GID4, with a KD value of 0.22 μM, and a ternary complex KD value of 2.85 μM. NEP108 can be utilized for cancer research.

Product Specifications

CAS Number

3031840-31-7

Smiles

CC=1C2=C (N3C ([C@H] (CC (NCCOCCOC=4C=C5C (=CC4) N=C (N5) [C@@H]6CC[C@H] (NC (CNCC7=CC=8C (N7) =CC=CC8) =O) CC6) =O) N=C2C9=CC=C (Cl) C=C9) =NN=C3C) SC1C