ERG-IN-4
ERG-IN-4 (Compound 12) is an orally active, selective ERG inhibitor with an IC50 value of 5.2 μM for hERG. It activates PXR and exhibits anticancer properties against non-small cell lung cancer lacking MTAP.
Product Specifications
CAS Number
3047672-14-7
Smiles
O=C (C=1C=CC=2N=C (N) C=3C=NN (C3C2C1) C) N (N (C (=O) C4CC4) C) CC5=NC=C (C=C5) C (F) (F) F
Molecular Formula
C24H22F3N7O2
Molecular Weight
497.48
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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