Desfluoro-BMS-694153
Desfluoro-BMS-694153 (Compound 3) is an antagonist of the calcitonin gene-related peptide receptor (CGRP receptor) with a Ki of 0.01 nM. It exhibits a significantly reduced risk of CYP3A4 inhibition, with IC50 values of 36 μM for CYP3A4-BFC and 6 μM for CYP3A4-BZR. Desfluoro-BMS-694153 is useful for migraine research.
Product Specifications
CAS Number
773886-89-8
Smiles
O=C1N (CC=2C (N1) =CC=CC2) C3CCN (C (N[C@H] (CC=4C=C5C (=C (C) C4) NN=C5) C (=O) N6CCC (CC6) N7CCCCC7) =O) CC3
Molecular Formula
C35H46N8O3
Molecular Weight
626.81
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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