PAR2 modulator-1
PAR2modulator-1 (Compound C781) is an antagonist of the protease-activated receptor 2 (PAR2) . It specifically inhibits the PAR2-dependent MAPK signaling pathway with an IC50 value of 8.5 μM. PAR2modulator-1 can effectively block pain responses triggered by PAR2 agonists. This compound is useful for research in inflammation, immunology, and neurological disorders, including chronic pain and asthma.
Product Specifications
CAS Number
2378159-28-3
Smiles
C (=O) (N1C2N ([C@@H] (CC (C) C) C (=O) N (CC3CCNCC3) C2) C (=O) [C@@H] (NC (CC (C) C) =O) C1) C4=CC=CO4
Molecular Formula
C27H41N5O5
Molecular Weight
515.66
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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