GRPR antagonist-3
GRPR antagonist-3 (compound (S) -1m) is a potent GRPR antagonist with an IC50 of 121 nM. It is stable in rat plasma and exhibits strong resistance to oxidative metabolism by microsomes in vitro. Additionally, GRPR antagonist-3 can be radiolabeled with fluorine-18 for use in PET imaging.
Product Specifications
CAS Number
2077238-49-2
Smiles
C (NC ([C@] (CC=1C=2C (NC1) =CC=CC2) (NC (NC3=CC=C (N (=O) =O) C=C3) =O) C) =O) C4 (CCCCC4) C5=CC=C (OCCF) C=N5
Molecular Formula
C33H37FN6O5
Molecular Weight
616.69
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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