RWT9996
RWT9996 acts as a balanced GPR17 antagonist. It inhibits G protein activation and β-arrestin-2 recruitment induced by MDL-29951. Additionally, RWT9996 suppresses MDL-29951-induced ERK/CREB phosphorylation and inositol phosphate (IP1) accumulation. This compound is useful for researching neurological disorders.
Product Specifications
CAS Number
2877694-62-5
Smiles
N#CC1=CC=C (NS (=O) (=O) C2=CNC (=C2) C=3C=CC=CC3) C (F) =C1
Molecular Formula
C17H12FN3O2S
Molecular Weight
341.36
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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