MKP10241
MKP10241 is an orally bioavailable GPR119 agonist that increases cAMP levels in GPR119-expressing cell lines with an EC50 of 3.7 nM. It significantly reduces blood glucose and glycated hemoglobin (HbA1c) levels in acute and chronic diabetic mouse models. It also exhibits favorable pharmacological activities in acute and chronic obesity models and MASH rodent models.
Product Specifications
CAS Number
2137977-29-6
Purity
99.79% (May vary between batches)
Smiles
FC1=C (C2=CN3C (=N2) SC (O[C@@H] (C) C4CCN (CC4) C=5N=CC (CC) =CN5) =N3) C=CC (S (C) (=O) =O) =C1
Molecular Formula
C24H27FN6O3S2
Molecular Weight
530.64
Storage Conditions
-20°C
Notes
For research use only.
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