5-HT4 antagonist 1
Product Specifications
UNSPSC Description
5-HT4 antagonist 1 is a 5-HT4 receptor antagonist with a pKi of 9.6.
Target Antigen
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein;Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/5-HT4_antagonist_1.html
Purity
98.67
Solubility
DMSO : 20 mg/mL (ultrasonic;warming;adjust pH to 3 with HCl;heat to 60°C)
Smiles
O=C(C1=C2OCCOC2=CC=C1)NCC3CCN(CCCS(=O)(N4CCN(C)CC4)=O)CC3
Molecular Weight
480.62
References & Citations
[1]Clark RD, et al. Identification of a 5-HT4 receptor antagonist clinical candidate through side-chain modification. Bioorg Med Chem Lett. 2005 Mar 15;15(6):1697-700.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-100170/5-HT4-antagonist-1-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-100170/5-HT4-antagonist-1-SDS-MedChemExpress.pdf
Clinical Information
No Development Reported
CAS Number
261766-73-8
Available Sizes
Curated Selection
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