TG-2-IN-4
TG-2-IN-4 (compound 8) is a transglutaminase 2 (TG2) inhibitor with an IC50 [1].
Product Specifications
CAS Number
[2410899-01-1]
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H335
Target
Glutaminase
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/tg-2-in-4.html
Purity
99.62
Solubility
DMSO : 125 mg/mL (ultrasonic)
Smiles
CC(C)CC1=C2C(N=C(N2)CN3C(C(NC([C@H](CC/C=C/C(N(C)C)=O)NC(OCC4=CC=CC=C4)=O)=O)=CC=C3)=O)=CC=C1
Molecular Formula
C34H40N6O5
Molecular Weight
612.72
Precautions
H302, H315, H319, H335
References & Citations
[1]Campbell D, et, al. Transglutaminase 2 (tg2) inhibitors. WO2020033784A1.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C, 3 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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