PSB-0963
PSB-0963 is a selective competitive extracellular 5'-nucleotidase (eN/CD73) inhibitor with a Ki value of 150 nM for rat extracellular 5'-nucleotidase. It exhibits greater selectivity compared to other extracellular nucleotidases (NTPDases 1-3) and P2Y receptors. PSB-0963 is applicable in cancer research.
Product Specifications
CAS Number
1213268-73-5
Field of Research
Immunology & Inflammation
Smiles
O=C1C2=C (C (C3=C (NC4=CC5=CC6=C (C=CC=C6) C=C5C=C4) C=C (S (=O) ([O-]) =O) C (N) =C13) =O) C=CC=C2.[Na+]
Molecular Formula
C28H17N2NaO5S
Molecular Weight
516.50
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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