What is the catalog number for NEP162?

The catalog number for NEP162 is orb3135971.

What sizes are available for NEP162?

NEP162 is available in the following size(s): 10 mg, 50 mg.

How many pack sizes does NEP162 come in?

NEP162 is available in 2 different pack sizes.

NEP162 is currently made to order / not held in immediate stock. Contact us for lead time.

NEP162

NEP162 is a BRD4 PROTAC degrader with DC50 values of 1.2 μM in SW480 cells and 1.6 μM in U2OS cells. NEP162 exhibits antiproliferative activity, effectively inhibiting tumor growth and inducing apoptosis. It is applicable in research on cancers such as osteosarcoma, colorectal cancer, and non-small cell lung cancer.

Product Specifications

CAS Number

3031840-36-2

Field of Research

Cell Biology, Epigenetics & Chromatin, Pharmacology & Drug Discovery

Smiles

CC=1C2=C (N3C ([C@H] (CC (=O) N4CCN (CCCOC=5C=C6C (=CC5) N=C (N6) [C@@H]7CC[C@H] (NC (CNCC8=CC=9C (N8) =CC=CC9) =O) CC7) CC4) N=C2C%10=CC=C (Cl) C=C%10) =NN=C3C) SC1C