TD-6301
TD-6301 is a bladder-selective M2/4 muscarinic receptor antagonist. It binds with high selectivity and blocks M2/4 muscarinic receptors, exhibiting particularly strong affinity for the human M2 receptor (Ki= 0.36 nM) . TD-6301 inhibits volume-induced bladder contraction (ID50= 0.075 mg/kg) and is applicable for studying overactive bladder conditions.
Product Specifications
CAS Number
690999-15-6
Field of Research
Neuroscience
Smiles
C (C (N) =O) ([C@H]1CN (CCCCCCCN (C (C) C) C2CCN (CC=3C (OC) =CC=NC3) CC2) CC1) (C4=CC=CC=C4) C5=CC=CC=C5
Molecular Formula
C40H57N5O2
Molecular Weight
639.91
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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