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DNMT-IN-5

DNMT-IN-5 is a potent and stable inhibitor of DNA methyltransferase (DNMT), with an IC50 of 0.78 nM. It exhibits submicromolar inhibitory activity against DNMT3A, upregulates the expression of target genes, inhibits cell proliferation, and induces key cell cycle arrest. DNMT-IN-5 is suitable for research on p53-deficient colorectal cancer.

Product Specifications

Field of Research

Epigenetics & Chromatin

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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