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DGK-IN-9

DGK-IN-9 (Compound 15) is an orally active and selective inhibitor of DGKζ with an IC50 of 6.1 nM. It is capable of activating IL-2 expression in Jurkat-IL2 nanoluc cells with an EC50 of 153 nM. DGK-IN-9 is applicable in tumor research.

Product Specifications

CAS Number

3081525-23-4

Field of Research

Immunology & Inflammation

Smiles

O=C (NC1=CC=C (OC=2C=CC=CC2F) C (=C1N (C) CCNC) C (F) (F) F) C3=NC (=CS3) C=4C=NN=CC4

Molecular Formula

C25H22F4N6O2S

Molecular Weight

546.54

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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