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TRPM8 antagonist 4 prodrug

TRPM8 antagonist 4 prodrug (Compound 8b) is an orally active CB2R agonist (EC50: 51.2 nM) and a weak TRPM8 antagonist. It acts as a prodrug of TRPM8 antagonist 4, exhibiting anti-inflammatory and analgesic properties. TRPM8 antagonist 4 prodrug is applicable in studies of inflammation-related pain disorders.

Product Specifications

Field of Research

Pharmacology & Drug Discovery, Pharmacology & Drug Discovery; Cell Biology

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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