BRD4-IN-10
BRD4-IN-10 (Compound 31) is a selective BRD4 inhibitor with an IC50 of 13.5 nM. It exhibits anti-inflammatory and anti-fibrotic effects, possesses good metabolic stability, favorable pharmacokinetic properties, and safety. BRD4-IN-10 is suitable for research in kidney fibrosis diseases.
Product Specifications
CAS Number
3051852-76-4
Field of Research
Epigenetics & Chromatin
Smiles
O=C1C2 (CCN (CC2) C3=NC (NC=4C=C5C (=CC4) N (C) C (=O) [C@@H] (C) N5C (C) C) =NC=C3) NC (=O) N1
Molecular Formula
C24H30N8O3
Molecular Weight
478.55
Storage Conditions
-20°C
Notes
For research use only.
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