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MRT-31619

MRT-31619 is a potent and selective CRBN degrader (MGD) that can degrade Cereblon (CRBN) . Its Ki value is 7.72 nM and its IC50 value is 14.1 nM. It can promote the dimerization of CRBN and lead to its degradation.

Product Specifications

Smiles

O=C (N1CCC2 (CN (C3=CC=C (CN (C4C (NC (CC4) =O) =O) C5=O) C5=C3) CC2) CC1) C6=CC=CC=C6

Molecular Formula

C28H30N4O4

Molecular Weight

486.57

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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