What is the catalog number for ETN029?

The catalog number for ETN029 is orb3134915.

What sizes are available for ETN029?

ETN029 is available in the following size(s): 25 mg, 50 mg, 100 mg.

How many pack sizes does ETN029 come in?

ETN029 is available in 3 different pack sizes.

ETN029 is currently made to order / not held in immediate stock. Contact us for lead time.

ETN029

ETN029 is a ligand targeting DLL3. The 225Ac-labeled ETN029 exhibits dose-dependent cytotoxic effects on small cell lung cancer (SCLC), neuroendocrine prostate cancer (NEPC), and metastatic melanoma cells, and can induce H2AX phosphorylation. The 177Lu-labeled ETN029 has rapid tumor uptake, sustained retention, and a favorable tumor-to-renal distribution ratio. Therefore, ETN029 can be used for imaging and mechanism studies of tumors such as SCLC and NEPC.

Product Specifications

CAS Number

3066864-32-9

Field of Research

Neuroscience, Protein Biochemistry, Stem Cell & Developmental Biology

Smiles

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