α2AR agonist 1
α2AR agonist 1 (compound S6a) is a morpholinopyrimidinone that serves as an agonist for the α2-adrenergic receptor (α2AR) . This compound elicits a concentration-dependent relaxation in precontracted aortic rings induced by phenylephrine (pEC50=6.81) . Additionally, α2AR agonist 1 elevates levels of NOx and NO in HUVEC.
Product Specifications
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Molecular Formula
C16H15N4NaO2
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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