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AR Degrader-1

AR Degrader-1 (Compound ML 2-9) is a monovalent degrader of androgen receptors (AR) categorized under molecular glues. In LNCaP prostate cancer cells, it facilitates AR degradation through DCAF16 (E3 ligase) while exhibiting minimal cytotoxicity.

Product Specifications

Field of Research

Metabolism Research, Pharmacology & Drug Discovery, Protein Biochemistry

Molecular Formula

C24H27ClN6O4S

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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