AR Degrader-1
AR Degrader-1 (Compound ML 2-9) is a monovalent degrader of androgen receptors (AR) categorized under molecular glues. In LNCaP prostate cancer cells, it facilitates AR degradation through DCAF16 (E3 ligase) while exhibiting minimal cytotoxicity.
Product Specifications
Field of Research
Metabolism Research, Pharmacology & Drug Discovery, Protein Biochemistry
Molecular Formula
C24H27ClN6O4S
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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