PAR4 antagonist 4
PAR4 antagonist4 (Compound 37) is a selective antagonist of protease-activated receptor 4 (PAR4) . It exhibits antiplatelet activity with an IC50 of 14.2 nM. Moreover, PAR4 antagonist3 enhances metabolic stability in human liver microsomes, showing a half-life (T1/2) of 42.5 minutes.
Product Specifications
CAS Number
3057206-41-1
Field of Research
Pharmacology & Drug Discovery
Smiles
FC1=CC=C (OCC2OC=3C=CC=4C=C (OC4C3OC2) C=5N=C6SC (=NN6C5) OC) C=C1
Molecular Formula
C22H16FN3O5S
Molecular Weight
453.44
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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