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IBG3

IBG3 is a bifunctional BET molecular glue degrader containing two JQ1 moieties, designed to target and degrade proteins through an intramolecular bivalent mechanism. It acts as a degrader for BRD2 and BRD4, with DC50 values of 8.6 pM and 6.7 pM, respectively.

Product Specifications

Field of Research

Epigenetics & Chromatin, Pharmacology & Drug Discovery

Molecular Formula

C54H57N9O5S2

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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