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Cbl-b-IN-16

Cbl-b-IN-16 (compound 31) is an orally active inhibitor of the RING E3 ligase Cbl-b, with an IC50 of 30 nM. It enhances IL-2 production in human T cells with an EC50 of 230 nM and exhibits antitumor activity.

Product Specifications

Field of Research

Cancer Biology, Protein Biochemistry

Molecular Formula

C26H27F3N6O

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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