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RXR agonist 1

RXR agonist 1 (Compound 33) is a highly selective RXR agonist, exhibiting EC50 values of 9 nM, 18 nM, and 11 nM for RXRα, RXRβ, and RXRγ, respectively. It demonstrates strong affinity for RXR with a Kd of 0.03 μM.

Product Specifications

Field of Research

Metabolism Research, Pharmacology & Drug Discovery

Molecular Formula

C18H20ClN3O3

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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