UPSEM792
UPSEM792 is a pharmacologically selective agonist molecule (PSEM) for PSAM4-GlyR, with an affinity Ki of 0.7 nM. It acts as a substrate for efflux transporters in both wild-type mice brains and in P-gp and BCRP double knockout mice. Additionally, uPSEM792 may serve as a lead compound in the development of PET radioligands for PSAM4-GlyR.
Product Specifications
CAS Number
2323525-19-3
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Smiles
O=C1C=NC=2C=C3C (=CC2N1C) C4CNCC3C4
Molecular Formula
C14H15N3O
Molecular Weight
241.29
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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